Write a note on Michaelis Menten equation for estimation of Km and Vmax.
[6 marks]Discuss causes of non - linearity with examples.
[4 marks]Write a note on Statistical moment theory.
[4 marks]Write a note on Mammillary and Catenary Model.
[6 marks]Discuss merits and demerits of non-compartmental pharmacokinetics.
[4 marks]Write a note on Physiological Pharmacokinetic model.
[4 marks]Define Bioavailability. Explain various methods used for determination of Bioavailability.
[6 marks]Write a note on elements of Bioavailability study protocol
[4 marks]Discuss Latin square design in Bioequivalent study
[4 marks]Define Drug Absorption. Enumerate various factors influencing GI absorption of a drug. Discuss Pharmaceutical factors in detail.
[6 marks]Discuss various barriers of Drug Distribution.
[4 marks]Explain Passive Diffusion in detail.
[4 marks]Explain One compartment open model for IV infusion.
[6 marks]Discuss the factors affecting renal excretion.
[4 marks]Define: (1) Peak plasma concentration (2) Area under the curve (3) Minimum effective Concentration (4) Duration of action Q. 6 (a) Explain Wagner Nelson method for computing absorption rate constant.
[6 marks]Explain two compartment open model for IV bolus administration.
[4 marks]Write a note on Apparent volume of distribution and its significance.
[4 marks]How Multiple dose regimen for IV bolus is determined?
[6 marks]How elimination rate can be determined using Urinary Excretion Data?
[4 marks]Describe any four methods to enhance the bioavailability through enhancement of Dissolution rate.
[4 marks]