Cl assify Sulfonamindes in detail with examples & structures.
[6 marks]Explain SAR activity of sulfonamides.
[5 marks]Write chemical name & synthesis of Sulfamethoxazole & Ofloxacin.
[5 marks]Classify fluoroquinolone & explain SAR activity of Fluoroquinolone.
[6 marks]Enlist different types of beta- lactum antibiotics with examples & structures & explain any one type in detail.
[5 marks]Classify Penicillin & explain mode of action of Penicillin.
[5 marks]Give any three structure of Macroliide antibiotics & explain why Arithromycin is unstable in acid media?
[6 marks]Explain SAR activity of Tetracyclines.
[5 marks]Explain chemical instability of penicillin in detail.
[5 marks]Classify anti malarial agents with examples & structures.
[6 marks]Explain SAR activity of aminoglycoside antibiotics.
[5 marks]Write chemical name & synthesis of Chloroquine & Metronidazole.
[5 marks]Explain XDR-TB. Write a note on second line anti TB agents.
[6 marks]Enlist with structure various azole anti fungal agents & explain mode of action of azole anti fungal agents.
[5 marks]Write chemical name & synthesis of Isoniazide & Ketoconazole. Q. 6 (a) Classify anti neoplastic agents with examples & structures.
[6 marks]Write a note on anti metabolites used as anti cancer agents.
[5 marks]Write a note on anti viral agents.
[5 marks]Explain in detail molecular modeling.
[6 marks]Write a note on methods of lead discovery.
[5 marks]Write a note on QSAR.
[5 marks]