Discuss in detail about various forces involved in drug receptor interactions.
[6 marks]Write short notes on DMARDs
[5 marks]Write chemical classification, mechanism of action, uses and side effect of Non-steroidal anti-inflammatory agents.
[5 marks]Briefly explain Phase 1 drug metabolism with examples.
[6 marks]Write short notes on factor affecting drug metabolism.
[5 marks]Write synthesis of Phenobarbitone and Phenytoin
[5 marks]Write SAR of Parasymapthomimetic agents.
[6 marks]Write SAR of acetylcholine antagonist.
[5 marks]Write synthesis of Adrenaline and Neostigmine
[5 marks]Write SAR of B-phenylehtanolamine adrenergic agonist.
[6 marks]Write detail notes on Neuromuscular junction blockers.
[5 marks]Write synthesis of Naphazoline and Salbutamol.
[5 marks]Briefly explain structural modification for Tricyclic Antidepressants.
[6 marks]Write detail SAR of Benzodiazepines derivatives.
[5 marks]Write synthesis of Fluoxetine and Imipramine. Q. 6 (a) Write SAR of Phenothazine derivatives.
[6 marks]Briefly explain structural modification of local anesthetic agents.
[5 marks]Write synthesis of Thiopental sodium and Lignocaine
[5 marks]Briefly explain Opiod Analgesics and Non-Opiod Analgesics. Write synthesis of Naproxen.
[6 marks]Write short details on below mentioned category:
[5 marks]Antiparkinson’s agent
[ marks]Anti-Alzheimer’s agent
[ marks]Explain analeptics and hallucinogens with examples.
[5 marks]