Describe USP dissolution apparatus with their application.
[6 marks]Explain physicochemical factors affecting GI absorption of drug.
[5 marks]Write a note on Passive diffusion.
[5 marks]Define: Pharmacokinetics, Clearance, Peak plasma concentration, Time of peak concentration, Area under curve, Therapeutic index.
[6 marks]Enlist extravascular routes for drug absorption. Discuss Topical route of administration.
[5 marks]Discuss physiological barriers for distribution of drugs.
[5 marks]Discuss significance of protein binding of drugs.
[6 marks]Discuss Wagner-Nelson method for estimation of Ka.
[5 marks]Enumerate different method for measurement of bioavailability. Discuss Pharmacokinetic methods for measurement of bioavailability.
[5 marks]Differentiate: compartment model and physiological model.
[6 marks]Describe factors affecting drug protein binding.
[5 marks]Write a note on Loading and maintenance dose.
[5 marks]Explain Michaelis-Menten Equation.
[6 marks]Discuss factors affecting renal clearance of drug.
[5 marks]Write a note on In-vitro - In-vivo correlations. Q. 6 (a) Define bioequivalence. Describe Latin square design for bioequivalence study.
[6 marks]Discuss Phase Ibiotransformation process.
[5 marks]Discuss causes of non-linearity with examples.
[5 marks]Explain methods for solubility enhancement of the drug.
[6 marks]Write note on Non compartmental Analysis.
[5 marks]Discuss open compartment model IV bolus administration
[5 marks]